Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,591
Tocris Bioscience™ SMER 3
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 67200-34-4 Molecular Formula: C11H4N4O2
| CAS | 67200-34-4 |
|---|---|
| Molecular Formula | C11H4N4O2 |
1,592
Tocris Bioscience™ DNQX
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CAS: 2379-57-9 Molecular Formula: C8H4N4O6
| CAS | 2379-57-9 |
|---|---|
| Molecular Formula | C8H4N4O6 |
1,593
Tocris Bioscience™ CU CPT 9a
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Potent TLR8 inhibitor
| CAS | 2165340-32-7 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2-Methyl-4-(7-methoxy-4-quinolinyl)phenol |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H15NO2 |
1,594
Tocris Bioscience™ PX 12
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CAS: 141400-58-0 Molecular Formula: C7H12N2S2
| CAS | 141400-58-0 |
|---|---|
| Molecular Formula | C7H12N2S2 |
1,595
Tocris Bioscience™ SB 366791
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CAS: 472981-92-3 Molecular Formula: C16H14ClNO2
| CAS | 472981-92-3 |
|---|---|
| Molecular Formula | C16H14ClNO2 |
1,597
Tocris Bioscience™ Tolvaptan
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Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
| Inhibitors | Tolvaptan |
|---|---|
| Product Type | Tolvaptan |
| Molecular Weight (g/mol) | 448.94 |
| Purity | >98% |
1,598
Tocris Bioscience™ TM2 TEAD inhibitor
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and reversible inhibitor of TEAD mediated Hippo/Yap signalling
| Target | YAP1 |
|---|---|
| CAS | 1008768-41-9 |
| Purity | 0.98 |
| Chemical Name or Material | 4-[3-(2-Cyclohexylethoxy)benzoyl]-N-phenyl-1-piperazinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C26H33N3O3 |
1,599
Tocris Bioscience™ Ki 20227
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 623142-96-1 Molecular Formula: C24H24N4O5S
| CAS | 623142-96-1 |
|---|---|
| Molecular Formula | C24H24N4O5S |
1,600
Tocris Bioscience™ A 410099.1
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High affinity XIAP antagonist
| Product Type | Antagonist |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H40N4O3.HCl |
| Formula Weight | 505.09 |
1,601
Tocris Bioscience™ CSN5i-3
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective CSN5 (COP9 signalosome) inhibitor
1,602
Tocris Bioscience™ GSK 2795039
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NADPH oxidase 2 (NOX2) inhibitor
| Target | NADPH Oxidase Inhibitors |
|---|---|
| CAS | 1415925-18-6 |
| Purity | 0.98 |
| Chemical Name or Material | N-[3-(2,3-Dihydro-1-methyl-1 H-indol-6-yl)-1-(1-methylethyl)-1 H-pyrrolo[2,3-b]pyridin-4-yl]-1-methyl-1 H-pyrazole-3-sulfonamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H26N6O2S |
1,603
Tocris Bioscience™ NVS PAK1 1
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Potent and selective PAK1 inhibitor
| CAS | 1783816-74-9 |
|---|---|
| Chemical Name or Material | (3S)-3-(2-Chloro-5-(2,2-difluoroethyl)-8-fluoro-5H-dibenzo[b,e][1,4]diazepin-11-ylamino)-N-isopropylpyrrolidine-1-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H25ClF3N5O |
| Formula Weight | Observed MW: 479.93 |
| Assay Percent Range | >98% |
1,604
Tocris Bioscience™ NVS PAK1 C
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Negative control of NVS PAK1 1
| Purity | 98% |
|---|---|
| Recommended Storage | Store at -20°C |
| Synonym | (3S)-3-(2-Chloro-5-(2,2-difluoroethyl)-8-fluoro-5H-dibenzo[b,e][1,4]diazepin-11-ylamino)-N,N-dimethylpyrrolidine-1-carboxamide |
| Molecular Formula | C22H23ClF3N5O |
| Formula Weight | 465.91 |
1,605
Tocris Bioscience™ L-NMMA acetate
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CAS: 53308-83-1 Molecular Formula: C9H20N4O4
| CAS | 53308-83-1 |
|---|---|
| Molecular Formula | C9H20N4O4 |